「Structural insights into the agonists binding and receptor selectivity of human histamine H₄ receptor」の関連論文
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Novel rearrangement reaction of morphinan derivatives and Design and synthesis of novel naphthalene-type orexin 2 receptor agonists
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Effect of Water Molecules on the Activating S810L Mutation of the Mineralocorticoid Receptor
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Redesigning the enzymatic synthetic pathway of adrenaline to produce non-natural compound, Phenylephrine [an abstract of entire text]
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Development of the first clinically used radiotracer [18F]T-401 for positron emission tomography imaging of monoacylglycerol lipase in brain (Monoacylglycerol lipase (MAGL)を標的としたPETトレーサー[18F]T-401の開発)
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Grafting Hydrophobic Amino Acids Critical for Inhibition of Protein–Protein Interactions on a Cell-Penetrating Peptide Scaffold
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医薬品候補の潜在的供給源としての野生塩生植物の利用
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硬骨魚類における補体成分C4アイソタイプの機能的多様性
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Discovery of Non-Cysteine-Targeting Covalent Inhibitors by Activity-Based Proteomic Screening with a Cysteine-Reactive Probe
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in vitroおよびin silico分析によるアディポネクチン受容体アゴニストジ・トリペプチドに関する研究
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Generation of molecular-targeting peptides for selective inhibition of the interaction between CTLA-4 and B7 in the dog: a new immune checkpoint inhibitor for cancer therapy
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Involvement of the γ isoform of cPLA₂ in the biosynthesis of bioactive N-acylethanolamines
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Mechanisms of anti-inflammatory and anticancer effects of biologically active components of cinobufacini
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Mode of Action Studies on Antitumor Macrolide Aplyronine A and Development of Actin-affinity Tags
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Transient Receptor Potential Vanilloid 1 アンタゴニストによるエネルギー代謝亢進作用に関する研究
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Promising SARS-CoV-2 main protease inhibitor ligand-binding modes evaluated using LB-PaCS-MD/FMO
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Immunostimulatory properties of CpG oligodeoxynucleotides forming monomeric guanine-quadruplex structure [an abstract of entire text]
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Mechanisms by which Bacterial and Viral Pathogens cause Ovarian dysfunction
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Self-assembling small-molecule adjuvants as antigen nano-carriers
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Increase of tissue factor expression on the surface of peripheral monocytes of patients with chronic spontaneous urticaria
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Increase of tissue factor expression on the surface of peripheral monocytes of patients with chronic spontaneous urticaria
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主要組織適合遺伝子複合体および血清アルブミンに対するリガンド分子による薬物送達効率の改善戦略
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Study on the regulation of CD8+ T cell immune response through nuclear receptor RORα and REV-ERB [an abstract of entire text]
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Oncogenic mutations Q61L and Q61H confer active form-like structural features to the inactive state (state 1) conformation of H-Ras protein
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Rocuronium Has a Suppressive Effect on Platelet Function via the P2Y12 Receptor Pathway In Vitro That Is Not Reversed by Sugammadex
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Identification of calcium and integrin-binding protein 1 (CIB1) as a novel regulator of production of Amyloid β peptide using CRISPR/Cas9-based screening system
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ニワトリにおけるTRPV1の酸感受性とその制御機構
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Magnetic Control of Cells by Chemical Fabrication of Melanin
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Dibromopinocembrin and Dibromopinostrobin Are Potential Anti-Dengue Leads with Mild Animal Toxicity
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Relationship among structure, cytotoxicity, and Michael acceptor reactivity of quinocidin
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Vaticanol C, a phytoalexin, induces apoptosis of leukemia and cancer cells by modulating expression of multiple sphingolipid metabolic enzymes
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Molecular basis for ANGPTL2 recognition of LILRB2 immune checkpoint receptor [an abstract of entire text]
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Allosteric regulation accompanied by oligomeric state changes of Trypanosoma brucei GMP reductase through cystathionine-β-synthase domain
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Studies on the Transport Mechanism and Physiological Roles of a Cargo Protein of Extracellular Membrane Vesicles from Shewanella vesiculosa HM13
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Endogenous agonist-bound S1PR3 structure reveals determinants of G protein-subtype bias
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Characterization of the Anticancer Activities of Some Natural and Synthetic Compounds: Molecular Targets and Mechanism
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Highly potent antiausterity agents from Callistemon species from Egypt and their mechanism of action against the PANC-1 human pancreatic cancer cell line
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Research for elucidation of immune evasion mechanisms and development of a novel immunotherapy for cancer in dogs [an abstract of entire text]
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Role of Persulfides/Polysulfides in Reversibility of S-Oxidation of Sensor Proteins during Oxidative Stress
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Suppression of Neuropeptide by Botulinum Toxin Improve Imiquimod-induced Psoriasis-like Dermatitis via the Regulation of Neuroimmune System
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Isolation of a human SARS-CoV-2 neutralizing antibody from a synthetic phage library and its conversion to fluorescent biosensors
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Studies on the prevention of influenza by vitamin D metabolite and vaccine in mice
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Study of the recognition of G-quadruplex DNA by human ORC protein
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Glycan Cluster Shielding and Antibody Epitopes on Lassa Virus Envelop Protein
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Design and synthesis of selective orexin 1 receptor antagonists with a morphinan skeleton and novel rearrangement reaction of morphinan skeleton
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A deazariboflavin chromophore kinetically stabilizes reduced FAD state in a bifunctional cryptochrome
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Observing the nonvectorial yet cotranslational folding of a multidomain protein, LDL receptor, in the ER of mammalian cells.
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Intramolecular Hydrofunctionalization Reactions of Alkenyl Amines Catalyzed by Disulfonimides
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Intramolecular Hydrofunctionalization Reactions of Alkenyl Amines Catalyzed by Disulfonimides
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Immunomodulatory effects of D-allose on cytokine production by plasmacytoid dendritic cells
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Immunomodulatory activity of phosphorylated buckwheat major allergen and its enzymatic hydrolysate (リン酸化ソバ主要アレルゲンとその酵素消化物の免疫調節作用)