「Xanthine derivatives inhibit FTO in an l-ascorbic acid-dependent manner」の関連論文
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Vaticanol C, a phytoalexin, induces apoptosis of leukemia and cancer cells by modulating expression of multiple sphingolipid metabolic enzymes
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Discovery of Bis-sulfonamides as Novel Inhibitors of Mitochondrial NADH-Quinone Oxidoreductase (Complex I)
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l-Asparaginase regulates mTORC1 activity via a TSC2-dependent pathway in pancreatic beta cells
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Discovery of Non-Cysteine-Targeting Covalent Inhibitors by Activity-Based Proteomic Screening with a Cysteine-Reactive Probe
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Role of Persulfides/Polysulfides in Reversibility of S-Oxidation of Sensor Proteins during Oxidative Stress
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アミノ酸およびペプチドによる食中毒細菌の生存とバイオフィルム形成の制御
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Natural tetramic acids elicit multiple inhibitory actions against mitochondrial machineries presiding over oxidative phosphorylation
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Bioactive Compounds Isolated from Celastrus hindsii B. and Associated Anti-gout, Anti-diabetic, and Anti-tyrosinase Potentials
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Dibromopinocembrin and Dibromopinostrobin Are Potential Anti-Dengue Leads with Mild Animal Toxicity
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Targeting tumor-intrinsic Nuclear Factor-kappa B signaling pathway for the discovery of anti-metastatic drug candidates from natural recourses
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The identification of novel small extracellular vesicle (sEV) production modulators using luciferase‐based sEV quantification method
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Lenalidomide derivatives and proteolysis-targeting chimeras for controlling neosubstrate degradation
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Identification of the ultrahigh-risk subgroup in neuroblastoma cases through DNA methylation analysis and its treatment exploiting cancer metabolism
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HDL promotes adiponectin gene expression via the CAMKK/CAMKIV pathway
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Studies on Histamine Production Properties and Control of Morganella psychrotolerans [an abstract of entire text]
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in vitroおよびin silico分析によるアディポネクチン受容体アゴニストジ・トリペプチドに関する研究
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Evaluation of Mongolian compound library for potential antimalarial and anti-Toxoplasma agents
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Characterization of the Anticancer Activities of Some Natural and Synthetic Compounds: Molecular Targets and Mechanism
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Inhibition of heat shock protein 90 destabilizes receptor tyrosine kinase ROR1 in lung adenocarcinoma
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医薬品候補の潜在的供給源としての野生塩生植物の利用
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ILF2 enhances the DNA cytosine deaminase activity of tumor mutator APOBEC3B in multiple myeloma cells
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Magnetic Control of Cells by Chemical Fabrication of Melanin
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ポリフェノールの食中毒細菌およびその毒素に対する作用機構に関する研究
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Development of the first clinically used radiotracer [18F]T-401 for positron emission tomography imaging of monoacylglycerol lipase in brain (Monoacylglycerol lipase (MAGL)を標的としたPETトレーサー[18F]T-401の開発)
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Carbonic anhydrase 9 confers resistance to ferroptosis/apoptosis in malignant mesothelioma under hypoxia
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Highly potent antiausterity agents from Callistemon species from Egypt and their mechanism of action against the PANC-1 human pancreatic cancer cell line
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Development of antisense oligonucleotides for suppressing breast cancer cell proliferation and the system for evaluating drug response of cardiomyocytes
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hMTH1阻害剤としての7,8-置換-デアザ-dGTP/dGMP 誘導体の合成と評価およびそれらのトリリン酸の細胞膜透過性の付与
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Redesigning the enzymatic synthetic pathway of adrenaline to produce non-natural compound, Phenylephrine [an abstract of entire text]
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An ACE2, SARS-CoV-2 spike protein binding protein, -like enzyme isolated from food-related microorganisms
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Pharmacologic characterization of TBP1901, a prodrug form of aglycone curcumin, and CRISPR-Cas9 screen for therapeutic targets of aglycone curcumin
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Effects of piperine, an active ingredient of white pepper, on growth, virulence expression and biofilm formation of Vibrio cholerae
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Generation of molecular-targeting peptides for selective inhibition of the interaction between CTLA-4 and B7 in the dog: a new immune checkpoint inhibitor for cancer therapy
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Luteolin suppress bladder cancer growth via regulation of mechanistic target of rapamycin (mTOR) pathway
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A simple method to distinguish residual elotuzumab from monoclonal paraprotein in immunofixation assays for multiple myeloma patients
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Chemical constituents and anti-pancreatic cancer activities of selected Thai medicinal plants
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Discovery of a Macropinocytosis‐Inducing Peptide Potentiated by Medium‐Mediated Intramolecular Disulfide Formation
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Sasa veitchii extract induces anticancer effects via inhibition of cyclin D1 expression in MCF-7 cells
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The mechanism of the conversion of alpha-eleostearic acid into conjugated linoleic acid
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植物ポリフェノールの抗菌および抗毒素活性に関する研究
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Enhanced G1 arrest and apoptosis via MDM4/MDM2 double knockdown and MEK inhibition in wild-type TP53 colon and gastric cancer cells with aberrant KRAS signaling
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高血圧自然発症ラットおよび血管内皮細胞におけるヘスペリジンの高血圧予防機構に関する研究
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Study of the Effects of Inhibition of Epigenetic Regulators on the Proliferation of Hematological Malignant Tumor Cells
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Promising SARS-CoV-2 main protease inhibitor ligand-binding modes evaluated using LB-PaCS-MD/FMO
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G-quadruplex-forming nucleic acids interact with splicing factor 3B subunit 2 and suppress innate immune gene expression
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Cathepsin K Activity Controls Cachexia-induced Muscle Atrophy via the Modulation of IRS1 Ubiquitination
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Antidepressant-like Effect and the Mechanism of Action of Lippia Citriodora Ethanolic Extract and Emulsion, and Verbascoside
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Inhibition of cyclooxygenase-1 by nonsteroidal anti-inflammatory drugs demethylates MeR2 enhancer and promotes Mbnl1 transcription in myogenic cells
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Nasturtium officinale Extract Suppresses Osteoclastogenesis in RAW 264 Cells by Inhibiting IκB-Kinase β
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Involvement of the γ isoform of cPLA₂ in the biosynthesis of bioactive N-acylethanolamines