「Elucidation of the Mechanism of Action of New Drug Candidates on Target Proteins」の関連論文
-
Ndufs4 ablation shows an elevated GFAP and a decreased synaptophysin expression in mouse hippocampus.
-
TDP-43 regulates cholesterol biosynthesis by inhibiting sterol regulatory element-binding protein 2
-
Epstein-Barr Virus BBLF1 Mediates Secretory Vesicle Transport to Facilitate Mature Virion Release
-
Oncogenic mutations Q61L and Q61H confer active form-like structural features to the inactive state (state 1) conformation of H-Ras protein
-
Biochemical, Cell Biological, and Molecular Dynamics Studies of the Fission Yeast α-Actinin Ain1
-
Internal dynamics of multidomain protein as revealed by an optimized neutron spin echo measurement and all-atom molecular dynamics simulation
-
A blast fungus zinc-finger fold effector binds to a hydrophobic pocket in host Exo70 proteins to modulate immune recognition in rice
-
Design and In vivo Evaluation of Novel mRNA Lipid Nanoparticles Beyond the Hepatocytes Towards a New Era of Personalized Gene Therapies [an abstract of entire text]
-
Synthesis and Molecular Docking of Bioactive Natural Products Containing (6H-Dibenzo[b,d]pyran-6-one) Framework.
-
A novel structural maintenance of chromosomes (SMC)-related protein family specific to Archaea
-
Study on the Pharmacological Effects of Organogermanium Compound THGP on RIG-I-Mediated Viral Sensing and Viral Replication during Influenza a Virus Infection
-
Identification and Characterization of Zn2+-Dependent DNAzymes
-
Combination of tumor necrosis factor-α and epidermal growth factor induces the adrenergic-to-mesenchymal transdifferentiation in SH-SY5Y neuroblastoma cells
-
MAGI-2 orchestrates the localization of backbone proteins in the slit diaphragm of podocytes
-
Family with sequence similarity 20 member B regulates osteogenic differentiation of bone marrow mesenchymal stem cells on titanium surfaces
-
Cleavage of TANK-Binding Kinase 1 by HIV-1 Protease Triggers Viral Innate Immune Evasion
-
Elucidation of the Regulatory Mechanism of Akt Activity and Investigation of Therapeutic Agents Focusing on the Pathway
-
Structure-based screening combined with computational and biochemical analyses identified the inhibitor targeting the binding of DNA Ligase 1 to UHRF1
-
Role of serotonin 4 receptor in the growth of axon and dendrites of hippocampal neurons during the embryonic development in mice
-
Time-resolved study on signaling pathway of photoactivated adenylate cyclase and its nonlinear optical response
-
Genetic dissection of resistance of two rice cultivars against blast fungus Magnaporthe oryzae
-
Cyclin J-CDK complexes limit innate immune responses by reducing proinflammatory changes in macrophage metabolism
-
Flavonoids and saponins in plant rhizospheres: roles, dynamics, and the potential for agriculture
-
Molecular basis for ANGPTL2 recognition of LILRB2 immune checkpoint receptor [an abstract of entire text]
-
Use of a Baculovirus-Mammalian Cell Expression-System for Expression of Drug-Metabolizing Enzymes: Optimization of Infection With a Focus on Cytochrome P450 3A4
-
Development studies based on Kampo theories for new treatment strategies and drug discoveries
-
Trimming gene deletion strategies for growth-coupled production in constraint-based metabolic networks: TrimGdel
-
Discovery of a phase-separating small molecule that selectively sequesters tubulin in cells
-
Effects of external molecular factors on the catalytic ability of bacterial RNase P ribozymes
-
Gut contractile organoids: a novel model system to study the cellular synchronization in gastrointestinal motility
-
Quantitative analysis of coordinated epithelial rotation on a two-dimensional discoidal pattern
-
Automated screening procedure for the phenotypes of congenital fibrinogen disorders using novel parameters, |min1|c and Ac/|min1|c, obtained from clot waveform analysis using the Clauss method
-
Modern Microscopic Approaches to Astrocytes
-
in vitroおよびin silico分析によるアディポネクチン受容体アゴニストジ・トリペプチドに関する研究
-
Comparison between the Light-Harvesting Mechanisms of Type-I Photosynthetic Reaction Centers of Heliobacteria and Photosystem I: Pigment Site Energy Distribution and Exciton State
-
hMTH1阻害剤としての7,8-置換-デアザ-dGTP/dGMP 誘導体の合成と評価およびそれらのトリリン酸の細胞膜透過性の付与
-
Bioactive Compounds Isolated from Celastrus hindsii B. and Associated Anti-gout, Anti-diabetic, and Anti-tyrosinase Potentials
-
リガンド支援型核磁気共鳴法による免疫賦活活性を持つ硫酸化多糖の分析評価に関する研究
-
Re-evaluation of the circadian clock model in mammals
-
Optimization of accelerator and brake in photosynthetic electron transport
-
Metabolic engineering of the l-serine biosynthetic pathway improves glutathione production in Saccharomyces cerevisiae
-
Immunoreactivity of urate transporters, GLUT9 and URAT1, is located in epithelial cells of the choroid plexus of human brains
-
Effects of piperine, an active ingredient of white pepper, on growth, virulence expression and biofilm formation of Vibrio cholerae
-
The accD3 gene for mycolic acid biosynthesis as a target for improving fatty acid production by fatty acid-producing Corynebacterium glutamicum strains
-
Immunoreactivity of receptor and transporters for lactate located in astrocytes and epithelial cells of choroid plexus of human brain
-
Development of perfluoroelastomer-based low-sorption microfluidic devices for drug metabolism and toxicity studies
-
Roles of TRPM4 in immune responses in keratinocytes and identification of a novel TRPM4-activating agent
-
Epigenomic dysregulation in AFP-producing gastric cancer
-
Electroanalysis for Quantitative Assessment of Bacterial Activity
-
Role of mitochondrial DNA damage in cigarette smoke extract-induced innate immunity and its clinical application to atherosclerosis screening